1. GPCR/G Protein
    Neuronal Signaling
  2. Adrenergic Receptor
  3. Tamsulosin

Tamsulosin (Synonyms: (R)-(-)-YM12617 free base; LY253351 free base)

Cat. No.: HY-B0661 Purity: 99.62%
Handling Instructions

Tamsulosin ((R)-(-)-YM12617 free base) is an inhibitor of α1-adrenergic receptor. Tamsulosin is used for the research of prostatic hyperplasia. Tamsulosin attenuates abdominal aortic aneurysm growth in animal models.

For research use only. We do not sell to patients.

Tamsulosin Chemical Structure

Tamsulosin Chemical Structure

CAS No. : 106133-20-4

Size Price Stock Quantity
Free Sample (0.5-1 mg)   Apply Now  
10 mM * 1 mL in DMSO USD 66 In-stock
Estimated Time of Arrival: December 31
10 mg USD 60 In-stock
Estimated Time of Arrival: December 31
50 mg USD 120 In-stock
Estimated Time of Arrival: December 31
100 mg USD 180 In-stock
Estimated Time of Arrival: December 31
200 mg   Get quote  
500 mg   Get quote  

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Customer Review

Based on 1 publication(s) in Google Scholar

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Description

Tamsulosin ((R)-(-)-YM12617 free base) is an inhibitor of α1-adrenergic receptor. Tamsulosin is used for the research of prostatic hyperplasia. Tamsulosin attenuates abdominal aortic aneurysm growth in animal models[1].

IC50 & Target[1]

α1-adrenergic receptor

 

Clinical Trial
Molecular Weight

408.51

Formula

C₂₀H₂₈N₂O₅S

CAS No.

106133-20-4

SMILES

O=S(C1=CC(C[[email protected]](NCCOC2=CC=CC=C2OCC)C)=CC=C1OC)(N)=O

Shipping

Room temperature in continental US; may vary elsewhere.

Storage
Powder -20°C 3 years
4°C 2 years
In solvent -80°C 6 months
-20°C 1 month
Solvent & Solubility
In Vitro: 

DMSO : 100 mg/mL (244.79 mM; Need ultrasonic)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.4479 mL 12.2396 mL 24.4792 mL
5 mM 0.4896 mL 2.4479 mL 4.8958 mL
10 mM 0.2448 mL 1.2240 mL 2.4479 mL
*Please refer to the solubility information to select the appropriate solvent.
In Vivo:
  • 1.

    Add each solvent one by one:  10% DMSO    40% PEG300    5% Tween-80    45% saline

    Solubility: ≥ 2.5 mg/mL (6.12 mM); Clear solution

  • 2.

    Add each solvent one by one:  10% DMSO    90% (20% SBE-β-CD in saline)

    Solubility: ≥ 2.5 mg/mL (6.12 mM); Clear solution

  • 3.

    Add each solvent one by one:  10% DMSO    90% corn oil

    Solubility: ≥ 2.5 mg/mL (6.12 mM); Clear solution

*All of the co-solvents are provided by MCE.
References
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This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

Keywords:

Tamsulosin(R)-(-)-YM12617LY253351LY 253351LY-253351Adrenergic ReceptorBeta Receptorprostatichyperplasiaaorticaneurysmabdominalreceptorsadrenergicalpha-1Inhibitorinhibitorinhibit

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Product Name:
Tamsulosin
Cat. No.:
HY-B0661
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