2. Signaling Pathways
  3. GPCR/G Protein
    Neuronal Signaling
  4. Dopamine Receptor
  5. D2 Receptor Isoform
  6. D2 Receptor Inhibitor

D2 Receptor Inhibitor

D2 Receptor Inhibitors (15):

Cat. No. Product Name Effect Purity
  • HY-10791
    Ritanserin
    		Inhibitor 99.78%
    Ritanserin (R 55667) is a highly potent, relatively selective, orally active, long acting antagonist of 5-HT2 receptor, with an IC50 of 0.9 nM, less active on Histamine H1, Dopamine D2, Adrenergic α1, Adrenergic α2 receptors.
  • HY-B0411
    Domperidone
    		Inhibitor 99.79%
    Domperidone (R33812) is an orally active and selective dopamine-2 receptor antagonist.
  • HY-B0520A
    Benztropine mesylate
    		Inhibitor 99.92%
    Benztropine mesylate (Benzatropine mesylate) is an orally active centrally acting anticholinergic agent that can be used for Parkinson's disease research.
  • HY-17390
    Loxapine
    		Inhibitor 99.69%
    Loxapine is an orally active dopamine inhibitor, 5-HT receptor antagonist and also a dibenzoxazepine anti-psychotic agent.
  • HY-B1904
    Fluphenazine decanoate
    		Inhibitor ≥98.0%
    Fluphenazine decanoate is a dopamine D2 receptor inhibitor, is a long-acting phenothiazine neuroleptic.
  • HY-B1262
    Acetophenazine dimaleate
    		Inhibitor 99.95%
    Acetophenazine dimaleate, a phenothiazine derivative, is an antipsychotic agent.
  • HY-17390A
    Loxapine succinate
    		Inhibitor 99.81%
    Loxapine succinate is an orally active dopamine inhibitor, 5-HT receptor antagonist and also a dibenzoxazepine anti-psychotic agent.
  • HY-B1196
    Tiapride hydrochloride
    		Inhibitor 99.82%
    Tiapride hydrochloride is a selective and orally active D2 and D3 dopamine receptors antagonist with IC50 values of 110-320 nM and 180 nM, respectively.
  • HY-B0901
    Bromperidol
    		Inhibitor 99.06%
    Bromperidol (R-11333) possesses antipsychotic activity, with a high affinity for central dopamine receptors D2.
  • HY-B0732
    Itopride hydrochloride
    		Inhibitor 99.85%
    Itopride (HSR803) hydrochloride is a potent dopamine-2 antagonist and an acetylcholine esterase (AChE) inhibitor.
  • HY-101622
    5-HT6/7 antagonist 1
    		Inhibitor
    5-HT6/7 antagonist 1 is a multifunctional ligand that antagonizes 5-HT6/7/2A and D2 receptors, without interacting with M1 receptors and hERG channels.
  • HY-17390B
    Loxapine hydrochloride
    		Inhibitor
    Loxapine hydrochloride is an orally active dopamine inhibitor, 5-HT receptor antagonist and also a dibenzoxazepine anti-psychotic agent.
  • HY-B0732A
    Itopride
    		Inhibitor
    Itopride (HSR803 free base) is a potent and orally active dopamine-2 antagonist and an acetylcholine esterase (AChE) inhibitor.
  • HY-116916
    Acetophenazine
    		Inhibitor
    Acetophenazine, a phenothiazine derivative, is an antipsychotic agent.
  • HY-B1904A
    Fluphenazine decanoate dihydrochloride
    		Inhibitor
    Fluphenazine decanoate dihydrochloride is a dopamine D2 receptor inhibitor, is a long-acting phenothiazine neuroleptic.