BET-IN-6
BET-IN-6 is a BET inhibitor. BET-IN-6 can be used as a Ligand for Target Protein for PROTAC for the synthesis of BRD2/BRD4 PROTAC degraders, such as PROTAC BRD2/BRD4 degrader-1 (HY-130612). BET-IN-6 can be used for cancer research.
For research use only. We do not sell to patients.
- CAS No.: 2570470-39-0
- Formula: C22H20N2O6S
- Molecular Weight:440.47
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
Description
IC50 & Target
[1]|
BRD4 |
BRD2 |
BET |
In Vitro
BET-IN-6 (Compound 24) is a BET inhibitor and can be used for the synthesis of PROTACs (Compounds 13-17)[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 2570470-39-0
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Molecular Weight 440.47
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Formula C22H20N2O6S
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SMILES
O=C(O)CCC1=CC2=C(C=CC(N(C3=O)C)=C2C3=C1)NS(=O)(C4=CC=CC=C4OC)=O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)