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Art. -Nr.: HY-185345

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GR119566X

GR119566X is a 5-HT₃ receptor ligand with a pK_i value of 8.80 against prufied 5-HT₃ receptor. GR119566X can be used for 5-HT₃ receptor purification.

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CAS. Nr.: 237752-42-0
Formel: C₂₀H₂₄N₄O
Molecular Weight:336.43

Speicherung:

Please store the product under the recommended conditions in the Certificate of Analysis.

GR119566X Chemical Structure

CAS. Nr.: 237752-42-0

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Beschreibung

GR119566X is a 5-HT₃ receptor ligand with a pK_i value of 8.80 against prufied 5-HT₃ receptor. GR119566X can be used for 5-HT₃ receptor purification^[1].

IC₅₀ & Target

5-HT₃ Receptor

Alle 5-HT Receptor Isoform-spezifische Produkte anzeigen :

In Vitro

GR119566X (12.5 mg; 16 h) is successfully coupled to Aﬃ-Gel 15 to form an affinity resin that specifically retains solubilized 5-HT₃ receptors from porcine cerebral cortex, enabling receptor purification^[1].
GR119566X (60 min at 37°C) binds to membrane-bound, solubilized, and affinity-purified 5-HT₃ receptors from porcine cerebral cortex with consistent high affinity, as shown by pK_i values ranging from 8.21 to 8.80^[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Chemical Information

CAS. Nr. 237752-42-0
Molecular Weight 336.43
Formel C₂₀H₂₄N₄O
SMILES

NCCCN1C(CCC(C2=O)CC3=C(N=CN3)C)=C2C4=C1C=CC=C4
Versand

Room temperature in continental US; may vary elsewhere.
Speicherung

Please store the product under the recommended conditions in the Certificate of Analysis.

Reinheit & Dokumentation

Handling Instructions (2659 KB)

Verweise

[1]. Fletcher S, et al. Purification of 5-hydroxytryptamine3 receptors from porcine brain. Br J Pharmacol. 1997 Oct;122(4):655-62. [Content Brief]

Calculators

Molaritätsrechner

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass Mass

Konzentration Konzentration

Volumen Volumen

Molecular Weight Molecular Weight

Verdünnungsrechner

Konzentration _{(Stammlösung)} × Volumen _{(Stammlösung)} = Konzentration _{(Ziellösung)} × Volumen _{(Ziellösung)}

Konzentration _{(Stammlösung)} Konzentration _{(Stammlösung)}

Volumen _{(Stammlösung)} Volumen _{(Stammlösung)}

Konzentration _{(Ziellösung)} Konzentration _{(Ziellösung)}

Volumen _{(Ziellösung)} Volumen _{(Ziellösung)}

Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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100 mg

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GR119566X

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Alle 5-HT Receptor Isoform-spezifische Produkte anzeigen

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GR119566X Related Classifications

HY-185345 Related Classifications