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Cat. No.: HY-116908

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SB-272183

SB-272183 is a selective 5-HT_1A, 5-HT_1B and 5-HT_1D receptor antagonist. In addition, SB-272183 is also a potent and selective ligand for 5-HT_1A, 5-HT_1B and 5-HT_1D receptors in human recombinant and native tissues with pK_i values of 8.0, 8.1 and 8.7, respectively. SB-272183 can be used in antidepressant research.

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CAS No.: 216058-27-4
화학식: C₂₉H₂₈ClN₅O
분자량:498.02

보관:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (270 KB)

SB-272183 Chemical Structure

CAS No.: 216058-27-4

Amount: USD 0.00

* 장바구니에 담기 전 물품의 수량을 선택해 주십시오.

Use of MCE Products

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Biological Activity
- 제품 설명
- IC₅₀ & Target
Chemical Information
순도&문서
References
Calculators
Help & FAQs
Classifications
Bioz

Biological Activity

제품 설명

IC₅₀ & Target

^[1]

5-HT_1A Receptor

5-HT_1B Receptor

5-HT_1D Receptor

5-HT_1A Receptor

8.0 (pKi)

5-HT_1B Receptor

8.1 (pKi)

5-HT_1D Receptor

8.7 (pKi)

All 5-HT Receptor Isoforms :

Chemical Information

CAS No. 216058-27-4
분자량 498.02
화학식 C₂₉H₂₈ClN₅O
SMILES

O=C(N1C2=CC(N3CCN(CC3)C)=C(C=C2CC1)Cl)NC4=C5C=CC=CC5=C(C6=CC=NC=C6)C=C4
선적

Room temperature in continental US; may vary elsewhere.
보관

Please store the product under the recommended conditions in the Certificate of Analysis.

순도&문서

Select Batch:

Purity: 99.98%

Assay: 99.98%

ee.: 99.98%

Data Sheet (270 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Handling Instructions (2659 KB)

References

[1]. Watson J, et al. SB‐272183, a selective 5‐HT1A, 5‐HT1B and 5‐HT1D receptor antagonist in native tissue[J]. British journal of pharmacology, 2001, 133(6): 797-806. [Content Brief]

Calculators

몰농도 계산기

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass Mass

Concentration Concentration

Volume Volume

Molecular Weight Molecular Weight

농도 희석 계산기

Concentration _(start) × Volume _(start) = Concentration _(final) × Volume _(final)

Concentration _(start) Concentration _(start)

Volume _(start) Volume _(start)

Concentration _(final) Concentration _(final)

Volume _(final) Volume _(final)

Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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MOQ

Minimum order quantity

100 mg

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Amount: USD 0.00

Biological Activity
- 제품 설명
- IC₅₀ & Target
Chemical Information
순도&문서
References

상품명:
Cat. No.:
수량:
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상품명:
CAS No.:
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Purity:
수량:

SB-272183

All 5-HT Receptor Isoforms

Biological Activity

제품 설명

IC50 & Target

Chemical Information

순도&문서

References

Calculators

Help & FAQs

SB-272183 Related Classifications

HY-116908 Related Classifications

Bioz

Keywords

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