MDL 27032
MDL 27032 is an active site-directed inhibitor of protein kinase C (PKC) and cAMP-dependent protein kinase (PKA) with Ki values of 24 and 14.3μM. MDL 27032 can relaxe vascular smooth muscle and can be used as vasodilator.
For research use only. We do not sell to patients.
- CAS No.: 110124-55-5
- Formula: C11H12N2O2
- Molecular Weight:204.23
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
Chemical Information
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CAS No. 110124-55-5
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Molecular Weight 204.23
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Formula C11H12N2O2
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SMILES
CCCC(N1)=C(C2=CC=NC=C2)OC1=O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
[1]. Robinson P J, et al. MDL 27,032 [4-propyl-5-(4-pyridinyl)-2 (3H)-oxazolone], an active site-directed inhibitor of protein kinase C and cyclic AMP-dependent protein kinase that relaxes vascular smooth muscle[J]. The Journal of pharmacology and experimental therapeutics, 1990, 255(3): 1392-1398. [Content Brief]
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
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