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Cat. No.: HY-145347

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GSK232

GSK232 is a highly selective, cellularly penetrant CECR2 inhibitor with excellent physicochemical properties.

For research use only. We do not sell to patients.

CAS No.: 2702984-69-6
Formula: C₂₁H₂₇ClN₆O₃S
Molecular Weight:479.00

Storage:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (267 KB)

GSK232 Chemical Structure

CAS No.: 2702984-69-6

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Use of MCE Products

Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Biological Activity

Description

GSK232 is a highly selective, cellularly penetrant CECR2 inhibitor with excellent physicochemical properties.

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Chemical Information

CAS No. 2702984-69-6
Molecular Weight 479.00
Formula C₂₁H₂₇ClN₆O₃S
SMILES

O=S(C(C=C1NC(CN2C3=C(CN(CC3)C)N=N2)=O)=C(C=C1)Cl)(N4C[C@@](C5CC5)([H])CC4)=O
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation

Select Batch:

Purity: 99.98%

Assay: 99.98%

ee.: 99.98%

Data Sheet (267 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Handling Instructions (2659 KB)

References

[1]. Lucas SCC, et al. Optimization of Potent ATAD2 and CECR2 Bromodomain Inhibitors with an Atypical Binding Mode. J Med Chem. 2020 May 28;63(10):5212-5241. [Content Brief]

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Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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100 mg

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GSK232

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Biological Activity

Chemical Information

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References

Calculators

Help & FAQs

GSK232 Related Classifications

HY-145347 Related Classifications