PARP1 degrader 1
PARP1 degrader 1 (Compound 2c) is a comparatively potent PARP1 HyT degrader (DC50: 618 nM for intracellular PARP-1). PARP1 degrader 1 is also a HyT-Olaparib (HY-10162) conjugate. PARP1 degrader 1 induces UPR/autophagy, thus facilitating the degradation of PARP-1. PARP1 Degrader 1 can be used in the research of cancer.
For research use only. We do not sell to patients.
- Formula: C42H42FN5O4
- Molecular Weight:699.81
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
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PARP-1 618 nM (DC50) |
Chemical Information
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Molecular Weight 699.81
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Formula C42H42FN5O4
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SMILES
O=C(N1CCN(CC1)C(C2=C(C=CC(CC3=NNC(C4=CC=CC=C43)=O)=C2)F)=O)CCCCNC(C5=CC=C(C=C5)C#CC#CC6CCCCC6)=O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
PARP1 degrader 1 Related Classifications
HY-180276 Related Classifications
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