PROTAC BRD4 Degrader-37
PROTAC BRD4 Degrader-37 (Compound TrimTAC-2) is a PROTAC BRD4 degrader. PROTAC BRD4 Degrader-37 has a DC50 of 36.4 nM and a Dmax of 73% in PANC-1 cells. PROTAC BRD4 Degrader-37 exhibits cytotoxicity against PANC-1 cells (GI50: 0.282 μM). PROTAC BRD4 Degrader-37 can be used in the research of tumors. (Pink: PROTAC BRD4 ligand-4 (HY-175242); Blue + Black: E3 ligase ligand + linker (HY-175241)).
For research use only. We do not sell to patients.
- Formula: C46H55N3O6S2
- Molecular Weight:810.08
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Biological Activity
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BRD4 |
Chemical Information
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Molecular Weight 810.08
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Formula C46H55N3O6S2
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SMILES
CSC1=CC=CC=C1C2=CC(S(C)(=O)=O)=C(C=C2)C(N(CC3CCCCC3)CCCCCCCNC(C4=CC5=C(C(C)=CC(C6=CN(C(C(C)=C6)=O)C)=C5)O4)=O)=O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
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