Tankyrase-IN-5
Tankyrase-IN-5 (Compound 30f), an analogue of MSC2504877 (HY-123851), is a tankyrase TNKS1 and TNKS2 inhibitor with IC50s of 2.3 nM and 7.9 nM, respectively.
For research use only. We do not sell to patients.
- CAS No.: 1460285-69-1
- Formula: C17H18N2O2
- Molecular Weight:282.34
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
IC50: 2.3 nM (TNKS1), 7.9 nM (TNKS2), 1900 nM (PARP1)[1]
Chemical Information
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CAS No. 1460285-69-1
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Molecular Weight 282.34
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Formula C17H18N2O2
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SMILES
O=C1NC(C2=CC=C(C(C)(C)O)C=C2)=CN3C=C(C)C=C13
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)