BET-IN-2
BET-IN-2 is a BET inhibitor with an IC50 of 52 nM for BRD4-BD1.
For research use only. We do not sell to patients.
- CAS No.: 2104688-91-5
- Formula: C23H29N3O
- Molecular Weight:363.50
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
|
BRD4 BD1 52 nM (IC50) |
|
Cell Line
|
Type | Value | Description | References |
|---|---|---|---|---|
| MM1.S | IC50 |
0.016 μM
Compound: 54
|
Antiproliferative activity against human MM1S cells after 72 hrs by CCK8 assay
Antiproliferative activity against human MM1S cells after 72 hrs by CCK8 assay
|
[PMID: 28586718] |
Chemical Information
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CAS No. 2104688-91-5
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Molecular Weight 363.50
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Formula C23H29N3O
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SMILES
CC1=C([C@H](C)NC2=CC(N(C3CC3)[C@H](C)C(N4C)=O)=C4C=C2)C=CC(C)=C1
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)