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  2. PI3K
  3. Umbralisib R-enantiomer

Umbralisib R-enantiomer (Synonyms: TGR-1202 R-enantiomer; RP5264 R-enantiomer)

Cat. No.: HY-12279F Purity: 99.52%
Handling Instructions

Umbralisib R-enantiomer (TGR-1202 R-enantiomer) is a PI3Kδ inhibitor, which is the less active enantiomer of TGR-1202.

For research use only. We do not sell to patients.

Umbralisib R-enantiomer Chemical Structure

Umbralisib R-enantiomer Chemical Structure

CAS No. : 1532533-69-9

Size Price Stock Quantity
10 mM * 1 mL in DMSO USD 1056 In-stock
Estimated Time of Arrival: December 31
2 mg USD 420 In-stock
Estimated Time of Arrival: December 31
5 mg USD 840 In-stock
Estimated Time of Arrival: December 31
10 mg   Get quote  
50 mg   Get quote  

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Customer Review

Based on 1 publication(s) in Google Scholar

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Description

Umbralisib R-enantiomer (TGR-1202 R-enantiomer) is a PI3Kδ inhibitor, which is the less active enantiomer of TGR-1202.

IC50 & Target

PI3Kδ

 

In Vitro

Umbralisib R-enantiomer (TGR-1202 R-enantiomer) (Formula A) exhibits a 50% inhibitory concentration (IC50) with respect to the δ type PI3-kinase that is at least 20-fold lower than the inhibitor's IC50 with respect to the rest of the other PI3K isoforms (i.e., a, β, and γ)[1].

Molecular Weight

571.55

Formula

C₃₁H₂₄F₃N₅O₃

CAS No.

1532533-69-9

SMILES

O=C1C(C2=CC=CC(F)=C2)=C([[email protected]@H](C)N3N=C(C4=CC=C(OC(C)C)C(F)=C4)C5=C(N)N=CN=C53)OC6=CC=C(F)C=C16

Shipping

Room temperature in continental US; may vary elsewhere.

Storage
Powder -20°C 3 years
  4°C 2 years
In solvent -80°C 6 months
  -20°C 1 month
References

Purity: 99.52%

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Keywords:

Umbralisib R-enantiomerTGR-1202 R-enantiomer RP5264 R-enantiomerPI3KPhosphoinositide 3-kinaseInhibitorinhibitorinhibit

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Umbralisib R-enantiomer
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HY-12279F
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