BAY-299 (Standard)
BAY-299 (Standard) is the analytical standard of BAY-299 (HY-107424). This product is intended for research and analytical applications. BAY-299, a chemical probe, is a very potent, dual inhibitor with IC50s of 67 nM for BRPF2 bromodomains (BD), 8 nM for TAF1 BD2, and 106 nM for TAF1L BD2.
For research use only. We do not sell to patients.
- CAS No.: 2080306-23-4
- Formula: C25H23N3O4
- Molecular Weight:429.47
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
IC50: 8 nM (TAF1 BD2), 106 nM (TAF1L BD2), 67 nM (BRPF2 BD), 3150 nM (BRPF1 BD), 5550 nM (BRPF3 BD)[1]
Chemical Information
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CAS No. 2080306-23-4
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Molecular Weight 429.47
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Formula C25H23N3O4
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SMILES
O=C(N1C2=C(C)C=C(N(C)C3=O)C(N3C)=C2)C4=CC=C(CCCO)C5=C4C(C1=O)=CC=C5
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)