BETi-211
BETi-211 is an orally active BET inhibitor (Ki: <1 nM). BETi-211 inhibits growth of triple-negative breast cancers (TNBC) cell lines with IC50 < 1 μM. BETi-211 degrades BET proteins and suppress tumor growth in xenograft breast tumors.
For research use only. We do not sell to patients.
- CAS No.: 1995867-02-1
- Formula: C26H29N7O3
- Molecular Weight:487.55
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
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BET |
Chemical Information
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CAS No. 1995867-02-1
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Molecular Weight 487.55
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Formula C26H29N7O3
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SMILES
COCC1=NC(NC2=CC(C3CC3)=NN2CC)=C4C(NC5=C4C=C(OC)C(C6=C(C)ON=C6C)=C5)=N1
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)