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Cat. No.: HY-143299

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BRD4-BD1-IN-1

BRD4-BD1-IN-1 (Compound 9a) is a BRD4-BD1 inhibitor with an IC₅₀ of 38.20 μM.

For research use only. We do not sell to patients.

CAS No.: 2761321-18-8
Formula: C₁₆H₁₅BrN₄O₄
Molecular Weight:407.22

Storage:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (272 KB)

BRD4-BD1-IN-1 Chemical Structure

CAS No.: 2761321-18-8

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Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Biological Activity
- Description
- IC₅₀ & Target
Chemical Information
Purity & Documentation
References
Calculators
Help & FAQs
Classifications
Bioz

Biological Activity

Description

BRD4-BD1-IN-1 (Compound 9a) is a BRD4-BD1 inhibitor with an IC₅₀ of 38.20 μM^[1].

IC₅₀ & Target

BRD4 BD1

38.20 μM (IC₅₀)

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Chemical Information

CAS No. 2761321-18-8
Molecular Weight 407.22
Formula C₁₆H₁₅BrN₄O₄
SMILES

CC(OCC1=NC2=C(N1CC3=CC(Br)=CC=C3)C(NC(N2C)=O)=O)=O
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation

Select Batch:

Purity: 99.98%

Assay: 99.98%

ee.: 99.98%

Data Sheet (272 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Handling Instructions (2659 KB)

References

[1]. Chang Y, et al. Design, synthesis, biological evaluation, and molecular docking of 1, 7-dibenzyl-substituted theophylline derivatives as novel BRD4-BD1-selective inhibitors. Medicinal Chemistry Research, 2021, 30(8): 1453-1468.

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Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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100 mg

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Biological Activity
- Description
- IC₅₀ & Target
Chemical Information
Purity & Documentation
References

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BRD4-BD1-IN-1

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Biological Activity

Chemical Information

Purity & Documentation

References

Calculators

Help & FAQs

BRD4-BD1-IN-1 Related Classifications

HY-143299 Related Classifications