1. Membrane Transporter/Ion Channel
    Neuronal Signaling
    GPCR/G Protein
    Metabolic Enzyme/Protease
  2. Calcium Channel
    mGluR
    Phosphodiesterase (PDE)
  3. CALP1 TFA

CALP1 TFA 

Cat. No.: HY-P1077A
Handling Instructions

CALP1 TFA is a calmodulin (CaM) agonist (Kd of 88 µM) with binding to the CaM EF-hand/Ca2+-binding site. CALP1 TFA blocks calcium influx and apoptosis (IC50 of 44.78 µM) through inhibition of calcium channel opening. CALP1 TFA blocks glutamate receptor channels and blocks a store-operated nonselective cation channel. CALP1 TFA activates CaM-dependent phosphodiesterase activity.

For research use only. We do not sell to patients.

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CALP1 TFA Chemical Structure

CALP1 TFA Chemical Structure

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Description

CALP1 TFA is a calmodulin (CaM) agonist (Kd of 88 µM) with binding to the CaM EF-hand/Ca2+-binding site. CALP1 TFA blocks calcium influx and apoptosis (IC50 of 44.78 µM) through inhibition of calcium channel opening. CALP1 TFA blocks glutamate receptor channels and blocks a store-operated nonselective cation channel. CALP1 TFA activates CaM-dependent phosphodiesterase activity[1][2][3][4].

IC50 & Target

Kd: 88 µM (Calmodulin)[4]

Molecular Weight

956.10

Formula

C₄₂H₇₆F₃N₉O₁₂

Sequence

Val-Ala-Ile-Thr-Val-Leu-Val-Lys

Sequence Shortening

VAITVLVK

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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Keywords:

CALP1CALP 1CALP-1Calcium ChannelmGluRPhosphodiesterase (PDE)Ca2+ channelsCa channelsMetabotropic glutamate receptorsCalmodulinEF-handcalciuminfluxglutamateInhibitorinhibitorinhibit

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CALP1 TFA
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HY-P1077A
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