1. GPCR/G Protein
    Immunology/Inflammation
  2. CCR
  3. CCR1 antagonist 9

CCR1 antagonist 9 

Cat. No.: HY-124759
Handling Instructions

CCR1 antagonist 9 is a potent and selective CCR1 antagonist with an IC50 of 6.8 nM in calcium flux assay.

For research use only. We do not sell to patients.

CCR1 antagonist 9 Chemical Structure

CCR1 antagonist 9 Chemical Structure

CAS No. : 1220026-26-5

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Description

CCR1 antagonist 9 is a potent and selective CCR1 antagonist with an IC50 of 6.8 nM in calcium flux assay[1].

IC50 & Target[1]

CCR1

6.8 nM (IC50, in calcium flux assay)

In Vitro

CCR1 antagonist 9 (Compound 19e) blocks the CCR1 chemotaxis of THP-1 cells with an IC50 of 28 nM. CCR1 antagonist 9 also blocks hERG with an IC50 of 30 μM[1].

Molecular Weight

425.44

Formula

C₂₀H₁₆FN₅O₃S

CAS No.

1220026-26-5

SMILES

O=C(C1=CN=CC2=C1C=NN2C3=CC=C(F)C=C3)NCC4=CC(S(=O)(C)=O)=NC=C4

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

References
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This equation is commonly abbreviated as: C1V1 = C2V2

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Keywords:

CCR1 antagonist 9CCRCC chemokine receptorCCR1autoimmuneinflammationChemokinereceptorsInhibitorinhibitorinhibit

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CCR1 antagonist 9
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