CPI-1328
CPI-1328 is an EZH2 inhibitor with a Ki value of 63 fM.
For research use only. We do not sell to patients.
- CAS No.: 2390367-27-6
- Formula: C28H36ClN3O4S
- Molecular Weight:546.12
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
All Histone Methyltransferase Isoforms
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Biological Activity
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EZH2 |
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Cell Line
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Type | Value | Description | References |
|---|---|---|---|---|
| HeLa | EC50 |
0.849 nM
Compound: 83
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Antiproliferative activity against human HeLa cells
Antiproliferative activity against human HeLa cells
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[PMID: 35531606] |
| KARPAS-422 | GI50 |
5.7 nM
Compound: 83
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Antiproliferative activity against human KARPAS-422 cells assessed as inhibition of cell growth
Antiproliferative activity against human KARPAS-422 cells assessed as inhibition of cell growth
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[PMID: 35531606] |
Chemical Information
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CAS No. 2390367-27-6
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Molecular Weight 546.12
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Formula C28H36ClN3O4S
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SMILES
ClC1=C2C(O[C@](O2)([C@]3([H])CC[C@H](CC3)N(C)C)C)=C(C4=C1CCN(C4=O)CC5=C(C=C(NC5=O)C)SC)C
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
CPI-1328 Related Classifications
HY-134899 Related Classifications
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