1. Metabolic Enzyme/Protease
  2. Phosphodiesterase (PDE)
  3. ent-Tadalafil

ent-Tadalafil (Synonyms: ent-IC-351)

Cat. No.: HY-90009C Purity: 97.42%
Handling Instructions

ent-Tadalafil (ent-IC-351), compound (6S,12aS), is a inactive cis-enantiomer of compound (6R,12aS). compound (6R,12aS) is a potent PDE5 inhibitor with an IC50 of 0.090 μM, while ent-Tadalafil is inactive at concentrations up to 10 µM.

For research use only. We do not sell to patients.

ent-Tadalafil Chemical Structure

ent-Tadalafil Chemical Structure

CAS No. : 629652-72-8

Size Price Stock Quantity
10 mM * 1  mL in DMSO USD 319 In-stock
Estimated Time of Arrival: December 31
5 mg USD 290 In-stock
Estimated Time of Arrival: December 31
10 mg USD 550 In-stock
Estimated Time of Arrival: December 31
50 mg   Get quote  
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Based on 1 publication(s) in Google Scholar

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Description

ent-Tadalafil (ent-IC-351), compound (6S,12aS), is a inactive cis-enantiomer of compound (6R,12aS). compound (6R,12aS) is a potent PDE5 inhibitor with an IC50 of 0.090 μM, while ent-Tadalafil is inactive at concentrations up to 10 µM[1].

IC50 & Target[1]

PDE5

10 μM (IC50)

Molecular Weight

389.40

Formula

C₂₂H₁₉N₃O₄

CAS No.

629652-72-8

SMILES

O=C([[email protected]]1([H])CC2=C([[email protected]](C3=CC=C(OCO4)C4=C3)N15)NC6=C2C=CC=C6)N(C)CC5=O

Shipping

Room temperature in continental US; may vary elsewhere.

Storage
Powder -20°C 3 years
  4°C 2 years
In solvent -80°C 6 months
  -20°C 1 month
References
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Keywords:

ent-Tadalafilent-IC-351Phosphodiesterase (PDE)cis-enantiomer6S,12aSInhibitorinhibitorinhibit

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