Etoperidone hydrochloride
Etoperidone hydrochloride, an antidepressant agent, is an orally active serotonin and nor-adrenaline re-uptake antagonist. Etoperidone hydrochloride shows Kd values of 36 nM, 38 nM, 85 nM, and 570 nM for 5-HT2 receptor, α1-adrenergic receptor, 5-HT1A receptor, and α2-adrenergic receptor, respectively.
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- CAS No.: 57775-22-1
- Formule: C19H29Cl2N5O
- Masse moléculaire:414.37
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Stockage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Activité biologique
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Chemical Information
- Pureté et documentation
- Références
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Help & FAQs
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Activité biologique
Description
IC50 & Target
[2]|
5-HT2 Receptor 36 nM (Kd) |
5-HT1A Receptor |
α1-adrenergic receptor 38 nM (Kd) |
5-HT1A Receptor 85 nM (Kd) |
α2-adrenergic receptor 570 nM (Kd) |
Chemical Information
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CAS No. 57775-22-1
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Masse moléculaire 414.37
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Formule C19H29Cl2N5O
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SMILES
O=C1N(CCCN2CCN(CC2)C3=CC(Cl)=CC=C3)N=C(CC)N1CC.Cl
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Livraison
Room temperature in continental US; may vary elsewhere.
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Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
[1]. B Cusack, et al. Binding of antidepressants to human brain receptors: focus on newer generation compounds. Psychopharmacology (Berl). 1994 May;114(4):559-65. [Content Brief]
[2]. G W Caldwell, et al. Evaluation of the absorption, excretion and metabolism of [14C] etoperidone in man. Xenobiotica. 2001 Nov;31(11):823-39. [Content Brief]
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Etoperidone hydrochloride Related Classifications
HY-106617A Related Classifications
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