FT001
Based on 1 Customer Validation
FT001 is an orally active and selective BET inhibitor. FT001 has potent anti-proliferative effects against MV-4-11. FT001 can be used for research of cancer.
For research use only. We do not sell to patients.
- Purity: 99.90%
- CAS No.: 1778655-51-8
- Formula: C25H29N3O4S
- Molecular Weight:467.58
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Storage:Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
Biological Activity
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Cell Line
|
Type | Value | Description | References |
|---|---|---|---|---|
| MV4-11 | GI50 |
0.22 μM
Compound: FT001
|
Growth inhibition of human MV411 cells after 72 hrs by Celltiter-Glo luminescent cell viability assay
Growth inhibition of human MV411 cells after 72 hrs by Celltiter-Glo luminescent cell viability assay
|
[PMID: 28835800] |
| NCT Number | Sponsor | Condition | Start Date |
Phase
|
|---|---|---|---|---|
| NCT01329991 | Plexxikon| | 2011-05 | PHASE1 |
Chemical Information
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CAS No. 1778655-51-8
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Appearance Solid
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Molecular Weight 467.58
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Formula C25H29N3O4S
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Color White to off-white
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SMILES
O=C(C1CC1)N2C3=CC(C4=CC=C(N5CCS(=O)(CC5)=O)C=C4)=CC=C3N([C@H](C2)C)C(C)=O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Powder -20°C 3 years 4°C 2 years In solvent -80°C 6 months -20°C 1 month
Purity & Documentation
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Data Sheet (268 KB)
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SDS (251 KB)
- English - EN (251 KB)
- Français - FR (251 KB)
- Deutsch - DE (251 KB)
- Norwegian - NO (251 KB)
- Español - ES (251 KB)
- Swedish - SV (251 KB)
- Italian - IT (251 KB)
- Portuguese - PT (251 KB)
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Handling Instructions (2659 KB)
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)