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MS453

MS453 is a potent and highly selective SETD8 inhibitor with an IC50 value of 804 nM. MS453 specifically modifies a cysteine residue close to the inhibitor binding site. MS453 is selective for 28 other methyltransferases. The crystal structure of MS453 reveals its binding mode to SETD8, providing an atomic-level view for the development of high-quality chemical probes for SETD8.

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  • CAS 番号: 2059892-29-2
  • 分子式: C20H27N5O3
  • 分子量:385.46
  • 保管条件:

    Please store the product under the recommended conditions in the Certificate of Analysis.

  • MS453 Chemical Structure
    MS453 構造式
CAS 番号: 2059892-29-2
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Histone Methyltransferase アイソフォーム固有の製品をすべて表示

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  • MS453 Chemical Structure
    MS453 Chemical Structure
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  • MS453