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Cat. No.: HY-186244

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Methyl-2-bromo-LSD

Name: Methyl-2-bromo-LSD
Brand: MedChemExpress
SKU: HY-186244
Price: 750.00 USD
Availability: InStock
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Methyl-2-bromo-LSD is a brain-penetrant 5-HT₂ receptor ligand. Methyl-2-bromo-LSD can be used for the research of alzheimer's disease, depression, schizophrenia, anxiety disorders.

For research use only. We do not sell to patients.

CAS No.: 50484-98-5
Formula: C₂₁H₂₆BrN₃O
Molecular Weight:416.35

Storage:

Please store the product under the recommended conditions in the Certificate of Analysis.

Methyl-2-bromo-LSD Chemical Structure

CAS No.: 50484-98-5

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Use of MCE Products

Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Biological Activity
- Description
- IC₅₀ & Target
- In Vivo
Chemical Information
Purity & Documentation
References
Calculators
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Biological Activity

Description

Methyl-2-bromo-LSD is a brain-penetrant 5-HT₂ receptor ligand. Methyl-2-bromo-LSD can be used for the research of alzheimer's disease, depression, schizophrenia, anxiety disorders^[1].

IC₅₀ & Target^[1]

5-HT₂ Receptor

All 5-HT Receptor Isoforms :

In Vivo

Methyl-2-bromo-LSD (0.1 μg/kg; i.v.; single dose) (as the stable component of [¹¹C]-MBL) selectively binds to serotonin 5-HT₂ receptors in baboon brain^[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Animal Model:

Papio anubis (adult male, 55 kg, anesthetized with Ketaset, 2% suritol, atropine)^[1]
Dosage:

0.1 μg/kg
Administration:

i.v.; single dose
Result:

Led to selective labeling of cortical brain regions, with highest activity in cortical areas and low activity in the cerebellum.
Showed significantly reduced cortical activity following ketanserin blockade.

Chemical Information

CAS No. 50484-98-5
Molecular Weight 416.35
Formula C₂₁H₂₆BrN₃O
SMILES

BrC1=C2C3=C(C=CC=C3C4=C[C@H](CN([C@@]4(C2)[H])C)C(N(CC)CC)=O)N1C
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation

Handling Instructions (2659 KB)

References

[1]. Wong DF, et al. Localization of serotonin 5-HT2 receptors in living human brain by positron emission tomography using N1-([11C]-methyl)-2-Br-LSD. Synapse. 1987;1(5):393-8.

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Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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Biological Activity
- Description
- IC₅₀ & Target
- In Vivo
Chemical Information
Purity & Documentation
References

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Methyl-2-bromo-LSD

All 5-HT Receptor Isoforms