PKi-402 (Standard)
PKi-402 (Standard) is the analytical standard of PKi-402 (HY-10683). This product is intended for research and analytical applications. PKi-402 is a selective, reversible, ATP-competitive inhibitor of PI3K, including PI3K-α mutants, and mTOR (IC50=2, 3, 7,14 and 16 nM for PI3Kα, mTOR, PI3Kβ, PI3Kδ and PI3Kγ).
For research use only. We do not sell to patients.
- CAS No.: 1173204-81-3
- Formula: C29H34N10O3
- Molecular Weight:570.65
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
IC50: 2 nM (PI3Kα), 3 nM (mTOR), 7 nM (PI3Kβ),14 nM (PI3Kδ), 16 nM (PI3Kγ)[1]
Chemical Information
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CAS No. 1173204-81-3
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Molecular Weight 570.65
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Formula C29H34N10O3
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SMILES
CCN1N=NC2=C1N=C(N=C2N3CCOCC3)C4=CC=C(C=C4)NC(NC5=CC=C(C=C5)C(N6CCN(CC6)C)=O)=O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)