1. Epigenetics
  2. Histone Methyltransferase
  3. SMYD2-IN-1

SMYD2-IN-1 is a SMYD2 inhibitor extracted from patent WO2016166186A1, compound example 1.1, has an IC50 of 4.45 nM.

For research use only. We do not sell to patients.

SMYD2-IN-1 Chemical Structure

SMYD2-IN-1 Chemical Structure

CAS No. : 2023788-96-5

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Description

SMYD2-IN-1 is a SMYD2 inhibitor extracted from patent WO2016166186A1, compound example 1.1, has an IC50 of 4.45 nM[1].

IC50 & Target

IC50: 4.45 nM (SMYD2)[1]

Molecular Weight

564.41

Formula

C25H25Cl2F2N7O2

CAS No.
SMILES

ClC1=CC(C2=NN(/C(NC3=CC=CC(OC(F)F)=C3)=N\C#N)CC2N(C([C@@H]4NCCC4)=O)CC)=CC=C1Cl

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation
References
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SMYD2-IN-1 Related Classifications

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The dilution calculator equation

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This equation is commonly abbreviated as: C1V1 = C2V2

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

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Product Name:
SMYD2-IN-1
Cat. No.:
HY-111810
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