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ZEN-3411 

Cat. No.: HY-111979
Handling Instructions

ZEN-3411 is a BET inhibitor with IC50s of 0.05, 0.05 and 0.06 μM for BRD4(BD1), BRD4(BD2) and BRD4(BD1BD2), respectively. ZEN-3411 can be used to form PROTACs to induce degradation of BRD4.

For research use only. We do not sell to patients.

ZEN-3411 Chemical Structure

ZEN-3411 Chemical Structure

CAS No. : 1952264-36-6

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Description

ZEN-3411 is a BET inhibitor with IC50s of 0.05, 0.05 and 0.06 μM for BRD4(BD1), BRD4(BD2) and BRD4(BD1BD2), respectively. ZEN-3411 can be used to form PROTACs to induce degradation of BRD4[1].

IC50 & Target[1]

BRD4 (BD1)

0.05 μM (IC50)

BRD4 (BD2)

0.05 μM (IC50)

BRD4(BD1BD2)

0.06 μM (IC50)

Molecular Weight

360.41

Formula

C₂₁H₂₀N₄O₂

CAS No.

1952264-36-6

SMILES

NC1=CC(C2=C(C)ON=C2C)=CC3=C1N=CN3CC4=CC=C(C5OC5)C=C4

Shipping

Room temperature in continental US; may vary elsewhere

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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ZEN-3411
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