1. Signaling Pathways
  2. Cytoskeleton
  3. Integrin
  4. α4β1 Inhibitors

α4β1 Inhibitors

αvβ1

αvβ3

αvβ5

αvβ6

αvβ8

α5β1

α1β1

α2β1

α4β1

α6β1

α9β1

αIIbβ3

α4β7

αLβ2

Your Search Returned No Results.

Sorry. There is currently no product that acts on isoform α4β1 together.

Please try each isoform separately.

α4β1 Specific Inhibitors, Agonists & Antagonists
Product Name α4β1 α5β1 α1β1 α2β1 α6β1 α9β1 αIIbβ3 α4β7 αLβ2 α4β1 Selectivity Purity
THI0019
α4β1, EC50: 1-2 μM
                Selective Agonist ≥98.0%
BIO5192
α4β1, IC50: 1.8 nM
   
α2β1, IC50: 1053 nM
 
α9β1, IC50: 138 nM
 
α4β7, IC50: >500 nM
  Selective Inhibitor
Integrin modulator 1
α4β1, IC50: 9.8 nM
                Selective Agonist 99.43%
Firategrast
α4β1
           
α4β7
  Selective Antagonist 99.88%
TR-14035
α4β1, IC50: 87 nM
           
α4β7, IC50: 7 nM
  Selective Antagonist 95.14%
BIO5192 hydrate
α4β1, IC50: 1.8 nM
   
α2β1, IC50: 1053 nM
 
α9β1, IC50: 138 nM
 
α4β7, IC50: >500 nM
  Selective Inhibitor ≥98.0%
Carotegrast methyl
α4β1
           
α4β7
  Selective Antagonist
BIO-1211
α4β1, IC50: 4 nM
α5β1, IC50: >100 μM
α1β1, IC50: >100 μM
 
α6β1, IC50: >100 μM
 
αIIbβ3, IC50: >100 μM
α4β7, IC50: 2 μM
αLβ2, IC50: >100 μM
Selective Inhibitor
BOP sodium
α4β1
       
α9β1
      Pan Inhibitor