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Tedizolid phosphate Chemical Structure
|Product name: Tedizolid phosphate|
|Cat. No.: HY-14855B|
Torezolid phosphate is a novel oxazolidinone for gram-positive infections, has an IC50 of 8.7 μM and 5.7 μM for monoamine oxidase (MAO)-A and MAO-B, respectively.
IC50 Value: 8.7 μM (MAO-A); 5.7 μM (MAO-B)
Tedizolid Phosphate is an oxazolidinone-class antibiotic. Tedizolid phosphate is a phosphate ester prodrug of the active compound tedizolid. It was developed for the treatment of acute bacterial skin and skin structure infections Tedizolid phosphate is a prodrug activated by plasma or intestinal phosphatases to tedizolid following administration of the drug either orally or intravenously. Once activated, tedizolid exerts its bacteriostatic microbial activity through inhibition of protein synthesis by binding to the 50S ribosomal subunit of the bacteria. Tedizolid phosphate was well tolerated following the oral administration of a once-daily 200-mg dose for three days.
|M.Wt||450.32||Storage||Please store the product under the recommended conditions in the Certificate of Analysis.|
|Solvent & Solubility||
DMSO: ≥ 36 mg/mL
|1 mg||5 mg||10 mg|
|1 mM||2.2206 mL||11.1032 mL||22.2064 mL|
|5 mM||0.4441 mL||2.2206 mL||4.4413 mL|
|10 mM||0.2221 mL||1.1103 mL||2.2206 mL|
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