ZEN-3411
ZEN-3411 is a BET inhibitor with IC50s of 0.05, 0.05 and 0.06 μM for BRD4(BD1), BRD4(BD2) and BRD4(BD1BD2), respectively. ZEN-3411 can be used to form PROTACs to induce degradation of BRD4.
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- CAS No.: 1952264-36-6
- Formule: C21H20N4O2
- Masse moléculaire:360.41
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Stockage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Activité biologique
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BRD4 (BD1) 0.05 μM (IC50) |
BRD4 (BD2) 0.05 μM (IC50) |
BRD4(BD1BD2) 0.06 μM (IC50) |
Chemical Information
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CAS No. 1952264-36-6
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Masse moléculaire 360.41
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Formule C21H20N4O2
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SMILES
NC1=CC(C2=C(C)ON=C2C)=CC3=C1N=CN3CC4=CC=C(C5OC5)C=C4
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Livraison
Room temperature in continental US; may vary elsewhere.
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Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)