1. Epigenetics
  2. Epigenetic Reader Domain
  3. CC-90010

CC-90010 

Cat. No.: HY-137573
Handling Instructions

CC-90010 (compound 1) is a reversible and orally active BET inhibitor. CC-90010 is applied in the study for advanced solid tumors.

For research use only. We do not sell to patients.

CC-90010 Chemical Structure

CC-90010 Chemical Structure

CAS No. : 1706738-98-8

Size Stock
10 mM * 1 mL in DMSO Check price and availability
5 mg Check price and availability
10 mg Check price and availability
50 mg Check price and availability
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Description

CC-90010 (compound 1) is a reversible and orally active BET inhibitor. CC-90010 is applied in the study for advanced solid tumors[1][2].

Molecular Weight

383.46

Formula

C₂₁H₂₁NO₄S

CAS No.

1706738-98-8

SMILES

O=C1N(C)C=C(C2=CC(S(=O)(C)=O)=CC=C2OCC3CC3)C4=C1C=CC=C4

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Solvent & Solubility
In Vitro: 

DMSO : 50 mg/mL (130.39 mM; Need ultrasonic)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.6078 mL 13.0392 mL 26.0783 mL
5 mM 0.5216 mL 2.6078 mL 5.2157 mL
10 mM 0.2608 mL 1.3039 mL 2.6078 mL
*Please refer to the solubility information to select the appropriate solvent.
In Vivo:
  • 1.

    Add each solvent one by one:  10% DMSO    90% corn oil

    Solubility: ≥ 2.08 mg/mL (5.42 mM); Clear solution

*All of the co-solvents are provided by MCE.
References
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The dilution calculator equation

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This equation is commonly abbreviated as: C1V1 = C2V2

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Keywords:

CC-90010CC90010CC 90010Epigenetic Reader DomainInhibitorinhibitorinhibit

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CC-90010
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