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Cat. No.: HY-108375

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CDK9 ligand-Linker Conjugate 1

CDK9 ligand-Linker Conjugate 1 is a compound formed by conjugation of a selective CDK9 ligand and a PROTAC linker. CDK9 ligand-Linker Conjugate 1 can be further coupled with an E3 ubiquitin ligase ligand to synthesize CDK9 PROTAC (HY-103628). CDK9 ligand-Linker Conjugate 1 is applicable to the research of CDK9-related disease states.

For research use only. We do not sell to patients.

CAS No.: 2118356-95-7
Formula: C₂₀H₂₆BrN₃O₂
Molecular Weight:420.34

Storage:

Please store the product under the recommended conditions in the Certificate of Analysis.

CDK9 ligand-Linker Conjugate 1 Chemical Structure

CAS No.: 2118356-95-7

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Use of MCE Products

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Biological Activity
- Description
- IC₅₀ & Target
Chemical Information
Purity & Documentation
References
Calculators
Help & FAQs
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Biological Activity

Description

IC₅₀ & Target^[1]

CDK9

All CDK Isoforms :

Chemical Information

CAS No. 2118356-95-7
Molecular Weight 420.34
Formula C₂₀H₂₆BrN₃O₂
SMILES

O=C(CC1=CC=C(OCCCCCBr)C=C1)NC2=CC(C3CCC3)=NN2
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation

Handling Instructions (2659 KB)

References

[1]. Robb CM, et al.. Chemically induced degradation of CDK9 by a proteolysis targeting chimera (PROTAC). Chemical communications (Cambridge, England). 2017 Jul 04;53(54):7577-7580. [Content Brief]

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Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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100 mg

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Biological Activity
- Description
- IC₅₀ & Target
Chemical Information
Purity & Documentation
References

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CDK9 ligand-Linker Conjugate 1

All CDK Isoforms