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Cat. No.: HY-149421

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BRD7-IN-3

BRD7-IN-3 (compound 1-78) is a dual inhibitor of bromodomain-containing proteins BRD7/BRD9 with IC₅₀s of 1.6 μM and 2.7 μM respectively.

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CAS No.: 3032601-04-7
Formule: C₁₈H₁₈N₂O₂
Masse moléculaire:294.35

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Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (267 KB)

BRD7-IN-3 Chemical Structure

CAS No.: 3032601-04-7

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Use of MCE Products

Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Activité biologique
- Description
- IC₅₀ & Target
Chemical Information
Pureté et documentation
Références
Calculators
Help & FAQs
Classifications
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Activité biologique

Description

BRD7-IN-3 (compound 1-78) is a dual inhibitor of bromodomain-containing proteins BRD7/BRD9 with IC₅₀s of 1.6 μM and 2.7 μM respectively^[1].

IC₅₀ & Target

IC50: 1.6 μM (BRD7), 2.7 μM (BRD9)^[1]

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Chemical Information

CAS No. 3032601-04-7
Masse moléculaire 294.35
Formule C₁₈H₁₈N₂O₂
SMILES

CC1=CC(N(C2=C1C=CC(C3=CC=C(N=C3C)OC)=C2)C)=O
Livraison

Room temperature in continental US; may vary elsewhere.
Stockage

Please store the product under the recommended conditions in the Certificate of Analysis.

Pureté et documentation

Select Batch:

Pureté: 99.98%

Assay: 99.98%

ee.: 99.98%

Fiche technique (267 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Instruction de manipulation (2659 KB)

Références

[1]. Ordonez-Rubiano SC, et al. Rational Design and Development of Selective BRD7 Bromodomain Inhibitors and Their Activity in Prostate Cancer. J Med Chem. 2023 Aug 24;66(16):11250-11270.. [Content Brief]

Calculators

Calculateur de molarité

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass Mass

Concentration Concentration

Volume Volume

Molecular Weight Molecular Weight

Calculateur de dilution

Concentration _(start) × Volume _(start) = Concentration _(final) × Volume _(final)

Concentration _(start) Concentration _(start)

Volume _(start) Volume _(start)

Concentration _(final) Concentration _(final)

Volume _(final) Volume _(final)

Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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100 mg

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- IC₅₀ & Target
Chemical Information
Pureté et documentation
Références

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BRD7-IN-3

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Activité biologique

Chemical Information

Pureté et documentation

Références

Calculators

Help & FAQs

BRD7-IN-3 Related Classifications

HY-149421 Related Classifications