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Cat. No.: HY-158051

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CIDD-0072424

CIDD-0072424 selectively inhibits Protein Kinase C-epsilon (PKCε) (K_i=54 nM). CIDD-0072424 reduces ethanol consumption and preference in a dose-dependent manner.

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CAS No.: 1620195-03-0
Formule: C₂₄H₂₉ClN₄O₂
Masse moléculaire:440.97

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Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (269 KB)

CIDD-0072424 Chemical Structure

CAS No.: 1620195-03-0

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Use of MCE Products

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

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- IC₅₀ & Target
Chemical Information
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Activité biologique

Description

CIDD-0072424 selectively inhibits Protein Kinase C-epsilon (PKCε) (K_i=54 nM). CIDD-0072424 reduces ethanol consumption and preference in a dose-dependent manner^[1].

IC₅₀ & Target

^[1]

PKCε

54 nM (Ki)

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Chemical Information

CAS No. 1620195-03-0
Masse moléculaire 440.97
Formule C₂₄H₂₉ClN₄O₂
SMILES

N[C@@H]([C@]1([H])CC[C@@](CC1)([H])C(NC2=CC=NC=C2)=O)CNC(C3(CC3)C4=CC=C(C=C4)Cl)=O
Livraison

Room temperature in continental US; may vary elsewhere.
Stockage

Please store the product under the recommended conditions in the Certificate of Analysis.

Pureté et documentation

Select Batch:

Pureté: 99.98%

Assay: 99.98%

ee.: 99.98%

Fiche technique (269 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Instruction de manipulation (2659 KB)

Références

[1]. De Kraker H, et al. Asymmetric Synthesis of CIDD-0072424 via an Enantioselective Nitro-Mannich Reaction: A Central Nervous System Penetrant, Selective Small Molecule Inhibitor of Protein Kinase C Epsilon. J Org Chem. 2024 Apr 5;89(7):5134-5141. [Content Brief]

Calculators

Calculateur de molarité

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass Mass

Concentration Concentration

Volume Volume

Molecular Weight Molecular Weight

Calculateur de dilution

Concentration _(start) × Volume _(start) = Concentration _(final) × Volume _(final)

Concentration _(start) Concentration _(start)

Volume _(start) Volume _(start)

Concentration _(final) Concentration _(final)

Volume _(final) Volume _(final)

Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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MOQ

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100 mg

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Chemical Information
Pureté et documentation
Références

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CIDD-0072424

Voir tous les produits spécifiques à Isoform PKC

Activité biologique

Description

IC50 & Target

Chemical Information

Pureté et documentation

Références

Calculators

Help & FAQs

CIDD-0072424 Related Classifications

HY-158051 Related Classifications

Bioz

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