JYL-79
JYL-79 is a TRPV1 agonist with the IC50 of 3.9 nM. JYL-79 can be used for study of neuropathic pain.
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- CAS No.: 289902-64-3
- Formule: C26H36N2O4S
- Masse moléculaire:472.64
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Stockage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Activité biologique
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Cell Line
|
Type | Value | Description | References |
|---|---|---|---|---|
| CHO | EC50 |
1.97 nM
Compound: 1
|
In vitro [Ca2+] influx relative to capsaicin by Rat Vanilloid receptor (VR1) expressing CHO cells
In vitro [Ca2+] influx relative to capsaicin by Rat Vanilloid receptor (VR1) expressing CHO cells
|
[PMID: 12825950] |
| CHO | EC50 |
1.97 nM
Compound: 2
|
Agonist activity at rat TRPV1 expressed in CHO cells assessed as maximal calcium uptake
Agonist activity at rat TRPV1 expressed in CHO cells assessed as maximal calcium uptake
|
[PMID: 17035013] |
Chemical Information
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CAS No. 289902-64-3
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Masse moléculaire 472.64
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Formule C26H36N2O4S
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SMILES
CC(C)(C)C(OCC(CNC(NCC1=CC=C(O)C(OC)=C1)=S)CC2=CC=C(C)C(C)=C2)=O
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Livraison
Room temperature in continental US; may vary elsewhere.
-
Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)