SEP-4199
SEP4199 is an orally active 5-HT7 receptor ligand, with a Ki value of 66 nM for human 5-HT7R and 16 nM for human D2R. SEP4199 mediates antidepressant effects. SEP4199 is applicable for the research of bipolar depression.
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- No. CAS: 2974362-88-2
- Fòrmula: C17H27N3O4S
- Peso molecular:369.48
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Almacenamiento:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Ver todos los productos específicos de isoformas 5-HT Receptor
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Actividad biológica
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D2 Receptor 16 nM (Ki) |
5-HT7 Receptor 66 nM (Ki) |
SEP4199 exhibits a higher relative affinity for human recombinant 5-HT7 receptors than human recombinant D2 receptors, with a 5-HT7R Ki of 66 ± 16 nM and a D2R Ki of 16 ± 0.62 nM[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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No. CAS 2974362-88-2
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Peso molecular 369.48
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Fòrmula C17H27N3O4S
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SMILES
CCN1[C@@H](CNC(C2=CC(S(=O)(CC)=O)=C(N)C=C2OC)=O)CCC1.CCN3[C@H](CNC(C4=CC(S(=O)(CC)=O)=C(N)C=C4OC)=O)CCC3
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Envío
Room temperature in continental US; may vary elsewhere.
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Almacenamiento
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureza y Documentación
Referencias
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
SEP-4199 Related Classifications
HY-14545B Related Classifications
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