MNI137
Based on 1 Customer Validation
MNI137 is a potent and selective negative allosteric modulator for group II mGluRs. MNI137 has IC50s values of 8.3 and 12.6 nM for human and rat mGlu2 inhibition of glutamate-induced calcium mobilization.
商品は「研究用試薬」です。人や動物の医療用・臨床診断用・食品用の製品ではありません。
研究用途以外に使用した場合、当社は一切の責任を負いかねます。
- 純度: 95.0%
- CAS 番号: 946619-21-2
- 分子式: C15H9BrN4O
- 分子量:341.16
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保管条件:Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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生物活性
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化学情報
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溶剤 & 溶解度
- 純度とドキュメンテーション
- 参考文献
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Help & FAQs
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生物活性
化学情報
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CAS 番号 946619-21-2
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性状 Solid
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分子量 341.16
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分子式 C15H9BrN4O
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Color Light brown to brown
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SMILES
N#CC1=NC=CC(C2=NC3=CC=C(Br)C=C3NC(C2)=O)=C1
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輸送条件
Room temperature in continental US; may vary elsewhere.
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保管条件
Powder -20°C 3 years 4°C 2 years In solvent -80°C 6 months -20°C 1 month
溶剤 & 溶解度
DMSO : 83.33 mg/mL (244.25 mM; ultrasonic and warming and heat to 60°C; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
濃度 (開始) × 体積 (開始) = 濃度 (終了) × 体積 (終了)
純度とドキュメンテーション
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データシート (269 KB)
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SDS (251 KB)
- English - EN (251 KB)
- Français - FR (251 KB)
- Deutsch - DE (251 KB)
- Norwegian - NO (251 KB)
- Español - ES (251 KB)
- Swedish - SV (251 KB)
- Italian - IT (251 KB)
- Korean - KR (251 KB)
- Portuguese - PT (251 KB)
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取扱説明書 (2659 KB)
参考文献
Complete Stock Solution Preparation Table
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
| Optional Solvent | Concentration Solvent Mass | 1 mg | 5 mg | 10 mg | 25 mg |
|---|---|---|---|---|---|
| DMSO | 1 mM | 2.9312 mL | 14.6559 mL | 29.3118 mL | 73.2794 mL |
| 5 mM | 0.5862 mL | 2.9312 mL | 5.8624 mL | 14.6559 mL | |
| 10 mM | 0.2931 mL | 1.4656 mL | 2.9312 mL | 7.3279 mL | |
| 15 mM | 0.1954 mL | 0.9771 mL | 1.9541 mL | 4.8853 mL | |
| 20 mM | 0.1466 mL | 0.7328 mL | 1.4656 mL | 3.6640 mL | |
| 25 mM | 0.1172 mL | 0.5862 mL | 1.1725 mL | 2.9312 mL | |
| 30 mM | 0.0977 mL | 0.4885 mL | 0.9771 mL | 2.4426 mL | |
| 40 mM | 0.0733 mL | 0.3664 mL | 0.7328 mL | 1.8320 mL | |
| 50 mM | 0.0586 mL | 0.2931 mL | 0.5862 mL | 1.4656 mL | |
| 60 mM | 0.0489 mL | 0.2443 mL | 0.4885 mL | 1.2213 mL | |
| 80 mM | 0.0366 mL | 0.1832 mL | 0.3664 mL | 0.9160 mL | |
| 100 mM | 0.0293 mL | 0.1466 mL | 0.2931 mL | 0.7328 mL |
MNI137 関連分類
HY-103572 関連分類
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