Milsaperidone
Milsaperidone ((S)-Hydroxy Iloperidone) is an active metabolite of the antipsychotic agent Iloperidone (HY-17410). Milsaperidone is a dopamine D2 and 5-HT2A receptor antagonist. Milsaperidone rapidly converts to Iloperidone when taken orally. Milsaperidone can be used in the research of mental illnesses such as depression.
For research use only. We do not sell to patients.
- CAS No.: 501373-88-2
- Formula: C24H29FN2O4
- Molecular Weight:428.50
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
| NCT Number | Sponsor | Condition | Start Date |
Phase
|
|---|---|---|---|---|
| NCT01329991 | Plexxikon| | 2011-05 | PHASE1 |
Chemical Information
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CAS No. 501373-88-2
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Molecular Weight 428.50
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Formula C24H29FN2O4
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SMILES
FC1=CC=C(C(C2CCN(CC2)CCCOC3=C(C=C(C=C3)[C@@H](O)C)OC)=NO4)C4=C1
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Synonyms
(S)-Hydroxy Iloperidone; VHX-896
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
[1]. Richmond L M. Med Check: FDA Accepts Bysanti Application, Cobenfy Fails as Adjunct, and More. 2025.
[2]. IsHak WW, et al. Depressive disorders: systematic review of approved psychiatric medications (2009-April 2025) and pipeline phase 3 medications. BMC Psychiatry. 2025 Oct 7;25(1):939. [Content Brief]
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)