1. PROTAC
    Epigenetics
  2. PROTAC
    Epigenetic Reader Domain
  3. PROTAC BET Degrader-10

PROTAC BET Degrader-10 

Cat. No.: HY-112718
Handling Instructions

PROTAC BET Degrader-10 is a potent BET protein BRD4 degrader extracted from patent WO2017007612A1, example 37, with a DC50 of 49 nM.

For research use only. We do not sell to patients.

PROTAC BET Degrader-10 Chemical Structure

PROTAC BET Degrader-10 Chemical Structure

CAS No. : 1957234-97-7

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Description

PROTAC BET Degrader-10 is a potent BET protein BRD4 degrader extracted from patent WO2017007612A1, example 37, with a DC50 of 49 nM[1].

Molecular Weight

783.29

Formula

C₃₉H₃₉ClN₈O₆S

CAS No.

1957234-97-7

SMILES

O=C(NCCCCCC(NCC1=CC=CC(C(N2C(CC3)C(NC3=O)=O)=O)=C1C2=O)=O)C[[email protected]]4C5=NN=C(C)N5C6=C(C(C)=C(C)S6)C(C7=CC=C(Cl)C=C7)=N4

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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Keywords:

PROTAC BET Degrader-10PROTAC BET Degrader10PROTAC BET Degrader 10PROTACEpigenetic Reader DomainProteolysis-targeting chimeraInhibitorinhibitorinhibit

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PROTAC BET Degrader-10
Cat. No.:
HY-112718
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