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Cat. No.: HY-118715

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Setin-1

Setin-1 is one of the most potent inhibitors of Set7, acting by inhibiting KMTase G9a.

For research use only. We do not sell to patients.

CAS No.: 1313802-67-3
Formula: C₂₉H₂₁F₃N₂O₂
Molecular Weight:486.48

Storage:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (269 KB)

Setin-1 Chemical Structure

CAS No.: 1313802-67-3

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Top Publications Citing

Use of MCE Products

Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Biological Activity

Description

Setin-1 is one of the most potent inhibitors of Set7, acting by inhibiting KMTase G9a^[1].

All Histone Methyltransferase Isoforms :

Chemical Information

CAS No. 1313802-67-3
Molecular Weight 486.48
Formula C₂₉H₂₁F₃N₂O₂
SMILES

FC(F)(C1=CC=C(C=C1)C2=CC=CC3=C2C=CN3C4=CC(CNC5=CC(C(O)=O)=CC=C5)=CC=C4)F
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation

Select Batch:

Purity: 99.98%

Assay: 99.98%

ee.: 99.98%

Data Sheet (269 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Handling Instructions (2659 KB)

References

[1]. Kashyap S, et al. Using 'biased-privileged' scaffolds to identify lysine methyltransferase inhibitors. Bioorg Med Chem. 2014 Apr 1;22(7):2253-60. [Content Brief]

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Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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100 mg

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Biological Activity
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Chemical Information
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References

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Setin-1

All Histone Methyltransferase Isoforms

Biological Activity

Chemical Information

Purity & Documentation

References

Calculators

Help & FAQs

Setin-1 Related Classifications

HY-118715 Related Classifications