TNKS-2-IN-4
TNKS-2-IN-4 (Compound 17) is a selective TNKS-2 inhibitor with an IC50 of 19 nM. TNKS-2-IN-4 exhibits anticancer activity against colorectal cancer.
For research use only. We do not sell to patients.
- CAS No.: 1613436-03-5
- Formula: C17H15NO
- Molecular Weight:249.31
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Biological Activity
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Chemical Information
- Protocols
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
Description
IC50 & Target
[1]|
TNKS2 19 nM (IC50) |
TNKS1 244 nM (IC50) |
PARP-1 860 nM (IC50) |
Chemical Information
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CAS No. 1613436-03-5
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Molecular Weight 249.31
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Formula C17H15NO
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SMILES
O=C1NC(C2=CC=CC=C2)=C(C)C3=C(C)C=CC=C31
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Protocols
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Cell Cytotoxicity Assay
Cytotoxicity assays are usually based on the assessment of cell membrane damage, which can also be indirectly detected by measuring cell viability. Detection methods include MTT assay, CKK-8 assay, LDH assay and ATP assay, etc.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
TNKS-2-IN-4 Related Classifications
HY-167762 Related Classifications
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