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ZEN-3219 

Cat. No.: HY-111977
Handling Instructions

ZEN-3219 is a BET inhibitor with IC50s of 0.48, 0.16 and 0.47 μM for BRD4(BD1), BRD4(BD2) and BRD4(BD1BD2), respectively. ZEN-3219 can be used to form PROTACs to induce degradation of BRD4.

For research use only. We do not sell to patients.

ZEN-3219 Chemical Structure

ZEN-3219 Chemical Structure

CAS No. : 1952264-34-4

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Description

ZEN-3219 is a BET inhibitor with IC50s of 0.48, 0.16 and 0.47 μM for BRD4(BD1), BRD4(BD2) and BRD4(BD1BD2), respectively. ZEN-3219 can be used to form PROTACs to induce degradation of BRD4[1].

IC50 & Target[1]

BRD4 (BD1)

0.48 μM (IC50)

BRD4 (BD2)

0.16 μM (IC50)

BRD4(BD1BD2)

0.47 μM (IC50)

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

References
Molecular Weight

322.36

Formula

C₁₉H₁₈N₂O₃

CAS No.

1952264-34-4

SMILES

O=C(C=CC(C1=C(C)ON=C1C)=C2)N2CC3=CC=C(C4OC4)C=C3

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Room temperature in continental US; may vary elsewhere

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Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

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Product Name:
ZEN-3219
Cat. No.:
HY-111977
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ZEN-3219

Cat. No.: HY-111977