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Cat. No.: HY-187059

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Piberaline

Name: Piberaline
Brand: MedChemExpress
SKU: HY-187059
Availability: PreOrder

(Synonyms: EGYT-475; Trelibet)

Piberaline (EGYT-475; Trelibet) is a psychoactive piperazine derivative with stimulant and antidepressant effects. Piberaline antagonizes Reserpine (HY-N0480)-induced dopamine depletion. Piberaline can be used for research on depression and central nervous system disorders.

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CAS No.: 39640-15-8
Formule: C₁₇H₁₉N₃O
Masse moléculaire:281.36

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Please store the product under the recommended conditions in the Certificate of Analysis.

Piberaline Chemical Structure

CAS No.: 39640-15-8

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Description

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In Vivo

Piberaline (EGYT-475; Trelibet) (up to 100 mg/kg; i.p.) showed no in vivo pharmacodynamic results in evaluated preclinical mouse studies^[1].
Piberaline is metabolized to produce N‑benzylpiperazine (BZP); the formed BZP can be further metabolized into 4′‑hydroxy‑BZP, 3′‑hydroxy‑BZP, 4′‑hydroxy‑3′‑methoxy‑BZP, piperazine, benzylamine and N‑benzylethylenediamine. Only 3‑4% of Piberaline is excreted into urine in the form of BZP^[3].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Chemical Information

CAS No. 39640-15-8
Masse moléculaire 281.36
Formule C₁₇H₁₉N₃O
SMILES

O=C(C1=NC=CC=C1)N2CCN(CC=3C=CC=CC3)CC2
Synonyms

EGYT-475; Trelibet
Livraison

Room temperature in continental US; may vary elsewhere.
Stockage

Please store the product under the recommended conditions in the Certificate of Analysis.

Pureté et documentation

Instruction de manipulation (2659 KB)

Références

[1]. D Dauzonne, et al. Synthesis and some CNS activities of new benzofuranylacryloylpiperazines,
European Journal of Medicinal Chemistry, Volume 30, Issue 1, 1995, Pages 53-59.

[2]. Nikonovich T, et al. Mechanochemical C–N Bond-Forming Reactions and Their Application in Pharmaceutical Synthesis. TalTech Press. 2024.

[3]. Staack RF, et al. Studies on the metabolism and toxicological detection of the new designer drug N-benzylpiperazine in urine using gas chromatography-mass spectrometry. J Chromatogr B Analyt Technol Biomed Life Sci. 2002 Jun 15;773(1):35-46.

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Piberaline

Voir tous les produits spécifiques à Isoform Dopamine Receptor

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