JYL-273
JYL-273 is a TRPV1 agonist, with the IC50 of 361 nM in CHO-TRPV1 cell lines.
Nur für Forschungszwecke. Wir verkaufen nicht an Patienten.
- CAS. Nr.: 1391826-17-7
- Formel: C28H39NO4S
- Molecular Weight:485.68
-
Speicherung:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
-
Biologische Aktivität
-
Chemical Information
- Reinheit & Dokumentation
- Verweise
-
Help & FAQs
Biologische Aktivität
361 nM (CHO-TRPV1 cell lines)[1].
|
Cell Line
|
Type | Value | Description | References |
|---|---|---|---|---|
| CHO | EC50 |
1.34 nM
Compound: 2
|
Agonist activity at human TRPV1 expressed in CHO cells assessed as 45Ca2+ uptake after 20 mins by liquid scintillation counting analysis
Agonist activity at human TRPV1 expressed in CHO cells assessed as 45Ca2+ uptake after 20 mins by liquid scintillation counting analysis
|
[PMID: 24321344] |
| CHO | EC50 |
2.83 nM
Compound: 2
|
In vitro [Ca2+] influx relative to capsaicin by Rat Vanilloid receptor (VR1) expressing CHO cells
In vitro [Ca2+] influx relative to capsaicin by Rat Vanilloid receptor (VR1) expressing CHO cells
|
[PMID: 12825950] |
Chemical Information
-
CAS. Nr. 1391826-17-7
-
Molecular Weight 485.68
-
Formel C28H39NO4S
-
SMILES
CC(C)(C)C(OCC(CC1=CC=C(C(C)(C)C)C=C1)CC(NCC2=CC=C(O)C(OC)=C2)=S)=O
-
Versand
Room temperature in continental US; may vary elsewhere.
-
Speicherung
Please store the product under the recommended conditions in the Certificate of Analysis.
Reinheit & Dokumentation
Verweise
Calculators
Konzentration (Stammlösung) × Volumen (Stammlösung) = Konzentration (Ziellösung) × Volumen (Ziellösung)
JYL-273 Related Classifications
HY-128479 Related Classifications
Powered by Bioz