DC-S100
DC-S100 is a potent SET7 inhibitor with an IC50 of 30.04 μM. DC-S100 binds to the cofactor (SAM) binding site of SET7 and forms hydrogen bonds and hydrophobic interactions with residues at this site. DC-S100 is applicable to biological studies of epigenetics and related diseases.
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- CAS No.: 178803-91-3
- Formule: C15H14N2O5
- Masse moléculaire:302.28
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Stockage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Activité biologique
Description
IC50 & Target
[1]|
SETD7/KMT7 30.04 μM (IC50) |
In Vitro
DC-S100 potently inhibits purified SET7 histone methyltransferase activity with an IC50 of 30.04 μM[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 178803-91-3
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Masse moléculaire 302.28
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Formule C15H14N2O5
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SMILES
O=C(C1=CC=C(C=C1)[N+]([O-])=O)NC2=CC=C(C(OC)=C2)OC
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Livraison
Room temperature in continental US; may vary elsewhere.
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Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)