JYL-273
JYL-273 is a TRPV1 agonist, with the IC50 of 361 nM in CHO-TRPV1 cell lines.
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- CAS No.: 1391826-17-7
- Formule: C28H39NO4S
- Masse moléculaire:485.68
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Stockage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Activité biologique
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Chemical Information
- Pureté et documentation
- Références
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Help & FAQs
Activité biologique
361 nM (CHO-TRPV1 cell lines)[1].
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Cell Line
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Type | Value | Description | References |
|---|---|---|---|---|
| CHO | EC50 |
1.34 nM
Compound: 2
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Agonist activity at human TRPV1 expressed in CHO cells assessed as 45Ca2+ uptake after 20 mins by liquid scintillation counting analysis
Agonist activity at human TRPV1 expressed in CHO cells assessed as 45Ca2+ uptake after 20 mins by liquid scintillation counting analysis
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[PMID: 24321344] |
| CHO | EC50 |
2.83 nM
Compound: 2
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In vitro [Ca2+] influx relative to capsaicin by Rat Vanilloid receptor (VR1) expressing CHO cells
In vitro [Ca2+] influx relative to capsaicin by Rat Vanilloid receptor (VR1) expressing CHO cells
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[PMID: 12825950] |
Chemical Information
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CAS No. 1391826-17-7
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Masse moléculaire 485.68
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Formule C28H39NO4S
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SMILES
CC(C)(C)C(OCC(CC1=CC=C(C(C)(C)C)C=C1)CC(NCC2=CC=C(O)C(OC)=C2)=S)=O
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Livraison
Room temperature in continental US; may vary elsewhere.
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Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
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