CSV0C018875
CSV0C018875 is a quinoline-based EHMT2/G9a inhibitor. CSV0C018875 exhibits lesser cytotoxicity than BIX-01294.
For research use only. We do not sell to patients.
- CAS No.: 442150-41-6
- Formula: C18H17ClN2O
- Molecular Weight:312.79
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
All Histone Methyltransferase Isoforms
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Biological Activity
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G9a |
CSV0C018875 (2.5-20 μM; 48 hours) inhibits the levels of H3K9me2 modifications in the histones[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
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Cell Line:HEK293 cells
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Concentration:2.5 μM, 10 μM, 20 μM
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Incubation Time:48 hours
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Result:Inhibited the enzymatic activity of G9a in a dose-dependent manner in HEK293 cells.
Chemical Information
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CAS No. 442150-41-6
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Molecular Weight 312.79
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Formula C18H17ClN2O
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SMILES
ClC(C=C1)=CC2=C1N=C(C)C=C2NC3=CC=C(OCC)C=C3
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
CSV0C018875 Related Classifications
HY-133031 Related Classifications
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