DC-S100
DC-S100 is a potent SET7 inhibitor with an IC50 of 30.04 μM. DC-S100 binds to the cofactor (SAM) binding site of SET7 and forms hydrogen bonds and hydrophobic interactions with residues at this site. DC-S100 is applicable to biological studies of epigenetics and related diseases.
For research use only. We do not sell to patients.
- CAS No.: 178803-91-3
- Formula: C15H14N2O5
- Molecular Weight:302.28
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
All Histone Methyltransferase Isoforms
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Biological Activity
Description
IC50 & Target
[1]|
SETD7/KMT7 30.04 μM (IC50) |
In Vitro
DC-S100 potently inhibits purified SET7 histone methyltransferase activity with an IC50 of 30.04 μM[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 178803-91-3
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Molecular Weight 302.28
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Formula C15H14N2O5
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SMILES
O=C(C1=CC=C(C=C1)[N+]([O-])=O)NC2=CC=C(C(OC)=C2)OC
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
DC-S100 Related Classifications
HY-125105 Related Classifications
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