DC-S100
DC-S100 is a potent SET7 inhibitor with an IC50 of 30.04 μM. DC-S100 binds to the cofactor (SAM) binding site of SET7 and forms hydrogen bonds and hydrophobic interactions with residues at this site. DC-S100 is applicable to biological studies of epigenetics and related diseases.
Para uso exclusivo en investigación. No vendemos a pacientes.
- No. CAS: 178803-91-3
- Fòrmula: C15H14N2O5
- Peso molecular:302.28
-
Almacenamiento:
Please store the product under the recommended conditions in the Certificate of Analysis.
Ver todos los productos específicos de isoformas Histone Methyltransferase
More
Actividad biológica
Descripciòn
IC50 & Target
[1]|
SETD7/KMT7 30.04 μM (IC50) |
In Vitro
DC-S100 potently inhibits purified SET7 histone methyltransferase activity with an IC50 of 30.04 μM[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
-
No. CAS 178803-91-3
-
Peso molecular 302.28
-
Fòrmula C15H14N2O5
-
SMILES
O=C(C1=CC=C(C=C1)[N+]([O-])=O)NC2=CC=C(C(OC)=C2)OC
-
Envío
Room temperature in continental US; may vary elsewhere.
-
Almacenamiento
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureza y Documentación
Referencias
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)