RL5a
Based on 1 Customer Validation
RL5a (compund C23) is a SETD8 inhibitor.
Para uso exclusivo en investigación. No vendemos a pacientes.
- Pureza : 99.60%
- No. CAS: 133671-66-6
- Fòrmula: C17H19N3O
- Peso molecular:281.35
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Almacenamiento:Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
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Actividad biológica
Descripciòn
IC50 & Target
SETD8[1]
Chemical Information
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No. CAS 133671-66-6
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Appearance Solid
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Peso molecular 281.35
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Fòrmula C17H19N3O
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Color Light yellow to light brown
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SMILES
CN(C)CCNC1=CC(C2=CC=CO2)=NC3=CC=CC=C13
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Envío
Room temperature in continental US; may vary elsewhere.
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Almacenamiento
Powder -20°C 3 years 4°C 2 years In solvent -80°C 6 months -20°C 1 month
Solvente y solubilidad
In Vitro:
DMSO : 40 mg/mL (142.17 mM; Need ultrasonic and warming; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Pureza y Documentación
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Ficha de datos (273 KB)
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SDS (251 KB)
- English - EN (251 KB)
- Français - FR (251 KB)
- Deutsch - DE (251 KB)
- Norwegian - NO (251 KB)
- Español - ES (251 KB)
- Swedish - SV (251 KB)
- Italian - IT (251 KB)
- Korean - KR (251 KB)
- Portuguese - PT (251 KB)
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Instrucciones de manejo (2659 KB)
Referencias
Complete Stock Solution Preparation Table
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
| Optional Solvent | Concentration Solvent Mass | 1 mg | 5 mg | 10 mg | 25 mg |
|---|---|---|---|---|---|
| DMSO | 1 mM | 3.5543 mL | 17.7715 mL | 35.5429 mL | 88.8573 mL |
| 5 mM | 0.7109 mL | 3.5543 mL | 7.1086 mL | 17.7715 mL | |
| 10 mM | 0.3554 mL | 1.7771 mL | 3.5543 mL | 8.8857 mL | |
| 15 mM | 0.2370 mL | 1.1848 mL | 2.3695 mL | 5.9238 mL | |
| 20 mM | 0.1777 mL | 0.8886 mL | 1.7771 mL | 4.4429 mL | |
| 25 mM | 0.1422 mL | 0.7109 mL | 1.4217 mL | 3.5543 mL | |
| 30 mM | 0.1185 mL | 0.5924 mL | 1.1848 mL | 2.9619 mL | |
| 40 mM | 0.0889 mL | 0.4443 mL | 0.8886 mL | 2.2214 mL | |
| 50 mM | 0.0711 mL | 0.3554 mL | 0.7109 mL | 1.7771 mL | |
| 60 mM | 0.0592 mL | 0.2962 mL | 0.5924 mL | 1.4810 mL | |
| 80 mM | 0.0444 mL | 0.2221 mL | 0.4443 mL | 1.1107 mL | |
| 100 mM | 0.0355 mL | 0.1777 mL | 0.3554 mL | 0.8886 mL |