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Referencia número: HY-168463

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Y16524

Y16524 is a potent inhibitor of CBP/p300 bromodomain , with the IC₅₀ of 0.01 μM. Y16524 has the potential for the research of acute myeloid leukemia (AML).

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No. CAS: 3109988-90-8
Fòrmula: C₃₀H₃₄ClN₅O₄
Peso molecular:564.08

Almacenamiento:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (273 KB)

Y16524 Chemical Structure

No. CAS: 3109988-90-8

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Use of MCE Products

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Actividad biológica

Descripciòn

Y16524 is a potent inhibitor of CBP/p300 bromodomain , with the IC₅₀ of 0.01 μM. Y16524 has the potential for the research of acute myeloid leukemia (AML)^[1].

Ver todos los productos específicos de isoformas Histone Acetyltransferase :

Ver todos los productos específicos de isoformas Epigenetic Reader Domain :

Chemical Information

No. CAS 3109988-90-8
Peso molecular 564.08
Fòrmula C₃₀H₃₄ClN₅O₄
SMILES

COC1=CC=C(N([C@H](C2=NC(C3=CC=C(ON=C4C)C4=C3)=CN2C[C@H](C)N5CCOCC5)CCC6)C6=O)C=C1Cl
Envío

Room temperature in continental US; may vary elsewhere.
Almacenamiento

Please store the product under the recommended conditions in the Certificate of Analysis.

Pureza y Documentación

Select Batch:

Pureza: 99.98%

Assay: 99.98%

ee.: 99.98%

Ficha de datos (273 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Instrucciones de manejo (2659 KB)

Referencias

[1]. Jian-Kang Hu, et al. Discovery of 5-imidazole-3-methylbenz[d]isoxazole derivatives as potent and selective CBP/p300 bromodomain inhibitors for the treatment of acute myeloid leukemia. Acta Pharmacol Sin. 2025 Jan 31. [Content Brief]

Calculators

Calculadora de molaridad

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass Mass

Concentration Concentration

Volume Volume

Molecular Weight Molecular Weight

Calculadora de dilución

Concentration _(start) × Volume _(start) = Concentration _(final) × Volume _(final)

Concentration _(start) Concentration _(start)

Volume _(start) Volume _(start)

Concentration _(final) Concentration _(final)

Volume _(final) Volume _(final)

Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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MOQ

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100 mg

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Actividad biológica
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Chemical Information
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Y16524

Ver todos los productos específicos de isoformas Histone Acetyltransferase

Ver todos los productos específicos de isoformas Epigenetic Reader Domain

Actividad biológica

Descripciòn

Chemical Information

Pureza y Documentación

Referencias

Calculators

Help & FAQs

Y16524 Related Classifications

HY-168463 Related Classifications

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